For research use only. Not for therapeutic Use.
Potent competitive vanilloid TRPV1 (VR1) receptor antagonist (IC<sub>50</sub> = 10 nM). Inhibits capsaicin-induced [Ca<sup>2+</sup>]<sub>i</sub> increase in rat DRG neurons, and guinea pig bladder and trachea contractions <em>in vitro</em>.
Catalog Number | I010484 |
CAS Number | 859171-97-4 |
Molecular Formula | C17H26INO3 |
Purity | ≥95% |
Target | TRP Channel |
Solubility | Soluble to 50 mM in ethanol and to 100 mM in DMSO |
Storage | Store at RT |
IUPAC Name | N-[(4-hydroxy-2-iodo-5-methoxyphenyl)methyl]nonanamide |
InChI | InChI=1S/C17H26INO3/c1-3-4-5-6-7-8-9-17(21)19-12-13-10-16(22-2)15(20)11-14(13)18/h10-11,20H,3-9,12H2,1-2H3,(H,19,21) |
InChIKey | AAORACFZMYMFCG-UHFFFAOYSA-N |
SMILES | CCCCCCCCC(=O)NCC1=CC(=C(C=C1I)O)OC |