Azatadine

• CAT Number: I003450
• CAS Number: 3964-81-6
• Molecular Formula: C20H22N2
• Molecular Weight: 290.4
• Purity: ≥95%
• Synonyms: 11-(1-methylpiperidin-4-ylidene)-5,6-dihydrobenzo[1,2]cyclohepta[3,4-b]pyridine
• Target: Histamine Receptor
• Solubility: 10 mM in DMSO
• Storage: Store at -20°C
• SMILES: CN1CCC(=C2C3=CC=CC=C3CCC4=C2N=CC=C4)CC1

Azatadine(Cat No.:I003450)is called 11-(1-methyl piperidine-4-ylidene)-5,6-dihydrobenzo[1,2]cyclohepta[3,4-b]pyridine.Azatadine is similar to cyproheptadine and has antihistamine, anticholinergic, anti-5-HT, and sedative effects. It is an inhibitor of the histamine receptor and choline receptor, with IC50 of 6.5 nM and 10 nM respectively.

Reference

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2: Togias AG, Naclerio RM, Warner J, Proud D, Kagey-Sobotka A, Nimmagadda I,
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