For research use only. Not for therapeutic Use.
BIM 23056, a linear octapeptide, is a potent sst3 and sst5 somatostatin receptor antagonist with Ki values of 10.8, 5.7, respectively[1].
BIM 23056 has Ki values of 142, 16.6, >1000 for sst1, sst4, sst2 , respectively[1].
Catalog Number | P000118 |
CAS Number | 150155-61-6 |
Molecular Formula | C71H81N11O9 |
Purity | ≥95% |
Reference | [1]. Y C Patel, et al. Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5). Endocrinology. 1994 Dec;135(6):2814-7. [2]. W Feniuk, et al. Further evidence from functional studies for somatostatin receptor heterogeneity in guinea-pig isolated ileum, vas deferens and right atrium. Br J Pharmacol. 1995 Jul;115(6):975-80. |