Bretylium tosylate

• CAT Number: I004331
• CAS Number: 61-75-6
• Molecular Formula: C18H24BrNO3S
• Molecular Weight: 414.36
• Purity: ≥95%
• Solubility: DMSO: ≥ 30 mg/mL
• Storage: Store at -20°C
• IUPAC Name: (2-bromophenyl)methyl-ethyl-dimethylazanium;4-methylbenzenesulfonate
• InChI: InChI=1S/C11H17BrN.C7H8O3S/c1-4-13(2,3)9-10-7-5-6-8-11(10)12;1-6-2-4-7(5-3-6)11(8,9)10/h5-8H,4,9H2,1-3H3;2-5H,1H3,(H,8,9,10)/q+1;/p-1
• InChIKey: KVWNWTZZBKCOPM-UHFFFAOYSA-M
• SMILES: CC[N+](C)(C)CC1=CC=CC=C1Br.CC1=CC=C(C=C1)S(=O)(=O)[O-]

 Bretylium (tosylate) (Cat.No:I004331) is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters. It is the sympathetic nerve and adrenergic ganglion blocking agent.   Bretylium tosylate inhibits adrenergic function presynaptically only after an initial release in neurotransmitter substance.   The reference for administration dose is 15 mg/kg.

Reference

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