For research use only. Not for therapeutic Use.
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.
| Catalog Number | I004341 |
| CAS Number | 620113-73-7 |
| Synonyms | (E)-2-(1,3-benzothiazol-2-yl)-3-[2-(4-fluorophenoxy)-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]prop-2-enenitrile |
| Molecular Formula | C25H15FN4O2S |
| Purity | ≥95% |
| InChI | InChI=1S/C25H15FN4O2S/c1-15-5-4-12-30-22(15)29-23(32-18-10-8-17(26)9-11-18)19(25(30)31)13-16(14-27)24-28-20-6-2-3-7-21(20)33-24/h2-13H,1H3/b16-13+ |
| InChIKey | IPZHFKHGSYRBNT-DTQAZKPQSA-N |
| SMILES | CC1=CC=CN2C1=NC(=C(C2=O)C=C(C#N)C3=NC4=CC=CC=C4S3)OC5=CC=C(C=C5)F |
| Reference | [1]. Levi L. Blazer et al.Reversible, Allosteric Small-Molecule Inhibitors of Regulator of G Protein Signaling Proteins. Molecular Pharmacology September 2010 vol.78 no.3 524-533 |
