For research use only. Not for therapeutic Use.
Selective ghrelin receptor (GhrR aka GHSR-1a) antagonist
| Catalog Number | I047596 |
| CAS Number | 2108806-12-6 |
| Molecular Formula | C25H33BrN4O3S.HCl |
| Purity | ≥95% |
| IUPAC Name | N-[(1R)-1-[3-[(4-bromophenyl)methyl]-1,2,4-oxadiazol-5-yl]-3-phenylpropyl]-3-(diethylamino)propane-1-sulfonamide;hydrochloride |
| InChI | InChI=1S/C25H33BrN4O3S.ClH/c1-3-30(4-2)17-8-18-34(31,32)29-23(16-13-20-9-6-5-7-10-20)25-27-24(28-33-25)19-21-11-14-22(26)15-12-21;/h5-7,9-12,14-15,23,29H,3-4,8,13,16-19H2,1-2H3;1H/t23-;/m1./s1 |
| SMILES | CCN(CC)CCCS(=O)(=O)N[C@H](CCC1=CC=CC=C1)C2=NC(=NO2)CC3=CC=C(C=C3)Br.Cl |
| Reference | KA Longo et al. Pharmacologic inhibition of ghrelin receptor signaling is insulin sparing and promotes insulin sensitivity. J. Pharmacol. Exp. Ther. 2011, 339(1), 115-124. |
