For research use only. Not for therapeutic Use.
CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
| Catalog Number | I002345 |
| CAS Number | 1802175-06-9 |
| Molecular Formula | C25H31N3O4 |
| Purity | ≥95% |
| Storage | 3 years-20°Cpowder |
| SMILES | CC1=CC(=C(C(=O)N1)CNC(=O)C2=C(N(C3=CC=CC=C32)C(C)C4CCOCC4)C)OC |
| Reference | [1] Bradley WD, et al. Chem Biol. 2014, 21(11), 1463-1475. |
