For research use only, not for therapeutic use.
Etravirine, also known as TMC 125 and R 165335, is a drug used for the treatment of HIV. Etravirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI). It was also approved in 2008. Etravirine, in combination with other anti-retrovirals, is indicated for the treatment of human immunodeficiency virus type 1 (HIV-1) infection in antiretroviral treatment-experienced adult patients, who have evidence of viral replication and HIV-1 strains resistant to a non-nucleoside reverse transcriptase inhibitor (NNRTI) and other antiretroviral agents.
Catalog Number | A000606 |
CAS Number | 269055-15-4 |
Synonyms | R-165335 |
Molecular Formula | C20H15BrN6O |
Purity | ≥95% |
Target | HIV |
Solubility | >19.4mg/mL in DMSO |
Storage | 3 years -20C powder |
InChIKey | PYGWGZALEOIKDF-UHFFFAOYSA-N |
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