For research use only. Not for therapeutic Use.
Felypressin(CAT: I004113) is a synthetic analog of vasopressin, acting as a selective agonist of the V1 vasopressin receptor. It exhibits strong vasoconstrictive properties, making it commonly used in dentistry to prolong the action of local anesthetics and reduce bleeding. Additionally, Felypressin is employed in pharmacological research to study vascular tone regulation and vasopressin receptor signaling pathways. Its targeted mechanism of action provides a valuable tool for exploring therapeutic approaches for conditions involving vascular dysfunction and hypotension.
Catalog Number | I004113 |
CAS Number | 56-59-7 |
Molecular Formula | C46H65N13O11S2 |
Purity | ≥95% |
Target | Vasopressin Receptor |
Solubility | DMSO ≥ 10.4 mg/mL |
Storage | -20°C |
IUPAC Name | (2S)-N-[(2S)-6-amino-1-[(2-amino-2-oxoethyl)amino]-1-oxohexan-2-yl]-1-[(4R,7S,10S,13S,16S,19R)-19-amino-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13,16-dibenzyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]pyrrolidine-2-carboxamide |
InChI | InChI=1S/C46H65N13O11S2/c47-18-8-7-14-29(40(64)52-23-38(51)62)54-45(69)35-15-9-19-59(35)46(70)34-25-72-71-24-28(48)39(63)55-31(20-26-10-3-1-4-11-26)43(67)56-32(21-27-12-5-2-6-13-27)42(66)53-30(16-17-36(49)60)41(65)57-33(22-37(50)61)44(68)58-34/h1-6,10-13,28-35H,7-9,14-25,47-48H2,(H2,49,60)(H2,50,61)(H2,51,62)(H,52,64)(H,53,66)(H,54,69)(H,55,63)(H,56,67)(H,57,65)(H,58,68)/t28-,29-,30-,31-,32-,33-,34-,35-/m0/s1 |
InChIKey | SFKQVVDKFKYTNA-DZCXQCEKSA-N |
SMILES | C1C[C@H](N(C1)C(=O)[C@@H]2CSSC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N2)CC(=O)N)CCC(=O)N)CC3=CC=CC=C3)CC4=CC=CC=C4)N)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N |