For research use only. Not for therapeutic Use.
GI-530159(Cat No.:I028033)is an investigational small molecule compound that acts as a selective positive allosteric modulator (PAM) of the γ-aminobutyric acid type A (GABA-A) receptor. It is designed to enhance GABAergic neurotransmission, which is involved in inhibitory signaling in the brain. GI-530159 has been studied for its potential neuropsychiatric applications, particularly for conditions such as anxiety, depression, and other disorders related to GABA dysfunction. By modulating GABA-A receptors, GI-530159 may offer a new approach to treat disorders involving neuronal excitability and imbalanced neurotransmission. Research is ongoing to evaluate its safety and efficacy.
Catalog Number | I028033 |
CAS Number | 69563-88-8 |
Synonyms | GI-530159, GI530159, GI 530159 |
Molecular Formula | C27H20F6N2O2 |
Purity | 98% |
Target | Potassium Channel |
Solubility | Soluble in DMSO |
Appearance | Solid powder |
Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
IUPAC Name | 4-[4-[2-[4-(4-aminophenoxy)phenyl]-1,1,1,3,3,3-hexafluoropropan-2-yl]phenoxy]aniline |
InChI | InChI=1S/C27H20F6N2O2/c28-26(29,30)25(27(31,32)33,17-1-9-21(10-2-17)36-23-13-5-19(34)6-14-23)18-3-11-22(12-4-18)37-24-15-7-20(35)8-16-24/h1-16H,34-35H2 |
InChIKey | HHLMWQDRYZAENA-UHFFFAOYSA-N |
SMILES | C1=CC(=CC=C1C(C2=CC=C(C=C2)OC3=CC=C(C=C3)N)(C(F)(F)F)C(F)(F)F)OC4=CC=C(C=C4)N |