GPR109 receptor agonist-2

• CAT Number: I040648
• CAS Number: 957129-38-3
• Molecular Formula: C7H10N2O2
• Molecular Weight: 154.17
• Purity: ≥95%
• Synonyms: 5-ethyl-4-methyl-1H-pyrazole-3-carboxylic acid
• InChI: InChI=1S/C7H10N2O2/c1-3-5-4(2)6(7(10)11)9-8-5/h3H2,1-2H3,(H,8,9)(H,10,11)
• InChIKey: MFNJGDMJKJLUGC-UHFFFAOYSA-N
• SMILES: CCC1=C(C(=NN1)C(=O)O)C

GPR109 receptor agonist-2 (Compound 5) is a selective GPR109a agonist with a pEC50 of 5.53[1].

Reference

[1]. Skinner PJ, et al. Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5620-3.
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