For research use only. Not for therapeutic Use.
Potent and highly selective histamine H<sub>3</sub> receptor agonist (pEC<sub>50</sub> = 9.74) that displays 300-fold selectivity over the H<sub>4</sub> receptor (pK<sub>i</sub> values are 9.07 and 6.61 respectively). Does not bind to H<sub>1</sub> or H<sub>2</sub> receptors at concentrations up to 10 <span class=/’symbol/’>μ</span>M.�.
Catalog Number | I010539 |
CAS Number | 699020-93-4 |
Synonyms | 4-(1H-Imidazol-4-ylmethyl)pyridine dihydrobromide |
Molecular Formula | C9H11Br2N3 |
Purity | ≥95% |
Target | Neuronal Signaling |
Solubility | Soluble to 100 mM in water |
Storage | Desiccate at RT |
IUPAC Name | 4-(1H-imidazol-5-ylmethyl)pyridine;dihydrobromide |
InChI | InChI=1S/C9H9N3.2BrH/c1-3-10-4-2-8(1)5-9-6-11-7-12-9;;/h1-4,6-7H,5H2,(H,11,12);2*1H |
InChIKey | CYNKWHIKNDIVDR-UHFFFAOYSA-N |
SMILES | C1=CN=CC=C1CC2=CN=CN2.Br.Br |