KN-93 Phosphate

• CAT Number: I011136
• CAS Number: 1188890-41-6
• Molecular Formula: C26 H29 Cl N2 O4 S . H3 O4 P
• Molecular Weight: 599.03
• Purity: ≥95%
• Storage: 3 years-20°Cpowder
• SMILES: CN(CC=CC1=CC=C(C=C1)Cl)CC2=CC=CC=C2N(CCO)S(=O)(=O)C3=CC=C(C=C3)OC.OP(=O)(O)O

KN-93 Phosphate is a potent and specific inhibitor of Ca2+/calmodulin-dependent protein kinase II (CaMKII) with Ki of 0.37 μM, no remarkable inhibitory effects on APK, PKC, MLCK or Ca2+-PDE activities. KN-93 attenuates CaMKII-induced autophagy.This product is not soluble in saline. Please do not dissolve it in saline for administration.

Reference

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