For research use only. Not for therapeutic Use.
Cytochrome P450 inhibitor. Inhibits several cytochrome P450 enzymes including aromatase (CYP19) and retinoic acid 4-hydroxylase (CYP26). Blocks retinoic acid metabolism (retinoic acid metabolism blocking agent, RAMBA). Displays antitumor activity against androgen-dependent and independent rat prostate carcinomas.
Catalog Number | I010609 |
Synonyms | Alternative Name: R-75251 |
Molecular Formula | C17H13ClN4.2HCl |
Purity | ≥95% |
Solubility | Soluble to 100 mM in DMSO and to 100 mM in water |
Storage | Desiccate at RT |