For research use only. Not for therapeutic Use.
Lirametostat (CPI-1205) is an orally available selective inhibitor of the histone lysine methyltransferase EZH2 with IC50 values of 2 nM and 52 nM for EZH2 and EZH1 respectively. It has potential antineoplastic activity.
| Catalog Number | I003555 |
| CAS Number | 1621862-70-1 |
| Molecular Formula | C27H33F3N4O3 |
| Purity | ≥95% |
| Storage | 3 years-20°Cpowder |
| SMILES | CC1=CC(=C(C(=O)N1)CNC(=O)C2=C(N(C3=CC=CC=C32)C(C)C4CCN(CC4)CC(F)(F)F)C)OC |
| Reference | [1] Vaswani RG, et al. J Med Chem. 2016. |
