MSP-3

• CAT Number: I011961
• CAS Number: 1820968-63-5
• Molecular Formula: C16H19NO3S
• Molecular Weight: 305.39
• Purity: ≥95%
• Synonyms: N-[(4-hydroxy-3-methoxyphenyl)methyl]-4-thiophen-2-ylbutanamide
• InChI: InChI=1S/C16H19NO3S/c1-20-15-10-12(7-8-14(15)18)11-17-16(19)6-2-4-13-5-3-9-21-13/h3,5,7-10,18H,2,4,6,11H2,1H3,(H,17,19)
• InChIKey: HCUVEUVIUAJXRB-UHFFFAOYSA-N
• SMILES: COC1=C(C=CC(=C1)CNC(=O)CCCC2=CC=CS2)O

MSP-3 is a potent TRPV1 agonist, with an EC50 of 0.87 μM. MSP-3 exhibits neuroprotective and antinociceptive effects[1].

Reference

[1]. Aiello F, et, al. Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl
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