Orphenadrine hydrochloride

• CAT Number: I003241
• CAS Number: 341-69-5
• Molecular Formula: C18H24ClNO
• Molecular Weight: 305.84
• Purity: ≥95%
• Target: Neuronal Signaling
• Solubility: 10 mM in H2O
• Storage: Store at -20°C
• IC50: 6.0 ±0.7 μM (Ki)

Orphenadrine hydrochloride (Cat.No:I003241) is a medication commonly used as a muscle relaxant to alleviate muscle spasms and associated pain. It acts by blocking certain nerve impulses responsible for muscle contractions. Orphenadrine hydrochloride is also prescribed for the symptomatic relief of Parkinson’s disease and is available in various formulations, including tablets and injections.

Reference

[1]. Kornhuber, J., et al., Orphenadrine is an uncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist: binding and patch clamp studies. J Neural Transm Gen Sect, 1995. 102(3): p. 237-46.
[2]. Pubill, D., et al., Assessment of the adrenergic effects of orphenadrine in rat vas deferens. J Pharm Pharmacol, 1999. 51(3): p. 307-12.