For research use only. Not for therapeutic Use.
CGP36742 is the first orally active GABAB-selective antagonist. CGP 36742/’s IC50 for blocking GABAergic transmission is 36 μM. CGP36742 in rats blocks baclofen-induced neuronal depression, and reduces learning deficit and passive avoidance in an olfactory bulbectomy depression model.
| Catalog Number | M135411 |
| CAS Number | 123690-78-8 |
| Molecular Formula | C7H18NO2P |
| Purity | ≥95% |
| Target | Neuronal Signaling |
| Storage | -20°C |
| IUPAC Name | 3-aminopropyl(butyl)phosphinic acid |
| InChI | InChI=1S/C7H18NO2P/c1-2-3-6-11(9,10)7-4-5-8/h2-8H2,1H3,(H,9,10) |
| InChIKey | ONNMDRQRSGKZCN-UHFFFAOYSA-N |
| SMILES | CCCCP(=O)(CCCN)O |
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