For research use only. Not for therapeutic Use.
GABAA agonist subtype α2 selective
Catalog Number | I009518 |
CAS Number | 205881-86-3 |
Molecular Formula | C23H20FN3O2 |
Purity | ≥95% |
IUPAC Name | 6-fluoro-9-methyl-2-phenyl-4-(pyrrolidine-1-carbonyl)pyrido[3,4-b]indol-1-one |
InChI | InChI=1S/C23H20FN3O2/c1-25-19-10-9-15(24)13-17(19)20-18(22(28)26-11-5-6-12-26)14-27(23(29)21(20)25)16-7-3-2-4-8-16/h2-4,7-10,13-14H,5-6,11-12H2,1H3 |
SMILES | CN1C2=C(C=C(C=C2)F)C3=C1C(=O)N(C=C3C(=O)N4CCCC4)C5=CC=CC=C5 |
Reference | G Griebel et al. SL651498: An Anxioselective Compound with Functional Selectivity for 2- and 3-Containing -Aminobutyric AcidA (GABAA) Receptors. J. Pharmaco. Eexp. Ther. 2001, 298(2), 753-768.
NR Mirza et al. Comparative cue generalisation profiles of L-838417, SL651498, zolpidem, CL218872, ocinaplon, bretazenil, zopiclone and various benzodiazepines in chlordiazepoxide and zolpidem drug discrimination. J. Ph. Exp. Ther. 2006, 316(3), 1291. |