For research use only. Not for therapeutic Use.
Tasipimidine sulfate is an orally active and selective α2A-adrenoceptor agonist with a pEC50 of 7.57 against human α2A-adrenoceptor. Tasipimidine sulfate can be used for situational anxiety and fear research[1].
| Catalog Number | I043598 |
| CAS Number | 1465908-73-9 |
| Synonyms | 2-(5-methoxy-3,4-dihydro-1H-isochromen-1-yl)-4,5-dihydro-1H-imidazole;sulfuric acid |
| Molecular Formula | C13H18N2O6S |
| Purity | ≥95% |
| InChI | InChI=1S/C13H16N2O2.H2O4S/c1-16-11-4-2-3-10-9(11)5-8-17-12(10)13-14-6-7-15-13;1-5(2,3)4/h2-4,12H,5-8H2,1H3,(H,14,15);(H2,1,2,3,4) |
| InChIKey | HZWPSPYSMWTZTG-UHFFFAOYSA-N |
| SMILES | COC1=CC=CC2=C1CCOC2C3=NCCN3.OS(=O)(=O)O |
| Reference | [1]. Lehtimäki J, et al. Tasipimidine-the pharmacological profile of a novel orally active selective α2A-adrenoceptor agonist. Eur J Pharmacol. 2022 May 15;923:174949. |
