For research use only. Not for therapeutic Use.
THIP (Gaboxadol) (Cat.No:I018297) is a selective δ-aminobutyric acid type A receptor (δ-GABAAR) agonist, functionally selective GABAAR ligand, exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GABAARs.
| Catalog Number | I018297 |
| CAS Number | 64603-91-4 |
| Molecular Formula | C₆H₈N₂O₂ |
| Purity | ≥95% |
| Reference | [1]. Hoestgaard-Jensen K, et al. Probing α4βδ GABAA receptor heterogeneity: differential regional effects of a functionally selective α4β1δ/α4β3δ receptor agonist on tonic and phasic inhibition in rat brain. J Neurosci. 2014 Dec 3;34(49):16256-72. |
