For research use only. Not for therapeutic Use.
TUG-1387 is a analog of both AH-7614 and TUG-1506 that has no activity at FFA4. TUG-1387 can serve as negative control for studies assessing FFA4 function.
| Catalog Number | M281235 |
| CAS Number | 6319-64-8 |
| Synonyms | 4-methyl-N-(9H-xanthen-9-yl)benzamide |
| Molecular Formula | C21H17NO2 |
| Purity | ≥95% |
| InChI | InChI=1S/C21H17NO2/c1-14-10-12-15(13-11-14)21(23)22-20-16-6-2-4-8-18(16)24-19-9-5-3-7-17(19)20/h2-13,20H,1H3,(H,22,23) |
| InChIKey | RWLHMQMVSKQATK-UHFFFAOYSA-N |
| SMILES | CC1=CC=C(C=C1)C(=O)NC2C3=CC=CC=C3OC4=CC=CC=C24 |
| Reference | [1]. Watterson KR, et al. Probe-Dependent Negative Allosteric Modulators of the Long-Chain Free Fatty Acid Receptor FFA4. Mol Pharmacol. 2017 Jun;91(6):630-641. [2]. Milligan G, et al. FFA4/GPR120: Pharmacology and Therapeutic Opportunities. Trends Pharmacol Sci. 2017 Sep;38(9):809-821. |
