UCPH 101

For research use only, not for therapeutic use.

  • CAT Number: I010767
  • CAS Number: 1118460-77-7
  • Molecular Formula: C27H22N2O3
  • Molecular Weight: 422.48
  • Purity: ≥95%
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UCPH 101(CAT: I010767) is a selective inhibitor of histone methyltransferase enhancer of zeste homolog 2 (EZH2). EZH2 is a key component of the polycomb repressive complex 2 (PRC2) and is involved in the epigenetic regulation of gene expression. UCPH 101 specifically targets the catalytic SET domain of EZH2, inhibiting its methyltransferase activity. By blocking EZH2-mediated histone methylation, UCPH 101 can potentially modulate gene expression patterns and have therapeutic implications in cancer and other diseases where dysregulation of EZH2 is implicated.


Catalog Number I010767
CAS Number 1118460-77-7
Synonyms

2-Amino-5,6,7,8-tetrahydro-4-(4-methoxyphenyl)-7-(naphthalen-1-yl)-5-oxo-4H-chromene-3-carbonitrile

Molecular Formula C27H22N2O3
Purity ≥95%
Solubility Soluble to 25 mM in DMSO
Storage Store at +4C

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