For research use only. Not for therapeutic Use.
A potent and selective inhibitor of the anandamide membrane transporter (AMT) with IC50 values of 4-11 μM. Displays negligible agonist activity at the hVR1 receptor and very weak action at CB1 and CB2 receptors. Ki values are 5-10 μM at CB1 and CB2. Active in vivo.
| Catalog Number | I010404 |
| CAS Number | 313998-81-1 |
| Synonyms | (5Z,8Z,11Z,14Z)-N-(4-Hydroxy-2-methylphenyl)-5,8,11,14-eicosatetraenamide |
| Molecular Formula | C27H39NO2 |
| Purity | ≥95% |
| Target | Cannabinoid Transporters |
| Solubility | Soluble in ethanol (supplied pre-dissolved in anhydrous ethanol, 5mg/ml) |
| Storage | Desiccate at -20°C |
| InChIKey | WUZWFRWVRHLXHZ-ZKWNWVNESA-N |
| SMILES | CCCCC/C=CC/C=CC/C=CC/C=CCCCC(=O)Nc1ccc(O)cc1C |
